Flupirtine Maleate 100 mg Description
Flupirtine maleate 100 mg is a non-opioid pain-relieving medication (analgesic) used for the treatment of moderate to severe acute pain.
What It Is
Flupirtine maleate is a centrally acting analgesic. It is not an opioid and does not belong to NSAIDs (like ibuprofen).
In some countries, it has been marketed under brand names such as Katadolon.
Important: Flupirtine has been restricted or withdrawn in several countries due to concerns about serious liver toxicity.
What It Is Used For
It has been prescribed for:
-
Musculoskeletal pain
-
Back pain
-
Post-operative pain
-
Cancer-related pain
-
Tension headaches
Usually intended for short-term use only.
How It Works
Flupirtine works by:
-
Opening neuronal potassium channels
-
Reducing excitability of nerve cells
-
Providing muscle-relaxant and pain-relieving effects
It also has mild NMDA receptor antagonist activity.
Tablet Description
-
Strength: 100 mg
-
Usually capsule-shaped or film-coated tablet
-
Often taken 23 times daily
-
Should be taken as directed by a doctor
-
Typically used for short durations (e.g., up to 2 weeks) due to liver risk
Common Side Effects
-
Dizziness
-
Drowsiness
-
Fatigue
-
Nausea
-
Dry mouth
Serious Warnings
Risk of liver damage (may cause hepatitis or liver failure).
Seek medical attention if you develop:
Avoid use in:
-
Patients with liver disease
-
People who consume heavy alcohol
-
Long-term therapy without monitoring